RegionInternational. Neutral scientific reference — not offered for sale here.
Cart · 0
Set region
Explore  /  VIP (Vasoactive Intestinal Peptide)
Research reference — not for sale

VIP (Vasoactive Intestinal Peptide)

A
lead outcome
Endogenous physiology (circadian/SCN,…
grades vary by outcome ↓
Peptide
also called — VIP · Vasoactive Intestinal Polypeptide
anti-inflammatory / immunoregulationcircadian (SCN)vasodilation / bronchodilationneuroprotection(gray-market: CIRS / mold-illness "capstone" therapy)

A profoundly important natural hormone — sold for a narrow, single-investigator gray-market niche. This entry is a study in contrast. Three threads: (1) VIP is a real endogenous neuropeptide with huge, well-established physiology — it's literally a master regulator of the brain's circadian clock; (2) yet its gray-market use is almost entirely one thing — a nasal spray in the "CIRS / mold-illness" protocol of a single physician (Ryan Shoemaker), where nearly all the human data come from that one investigator; (3) the honest gap between "fundamentally important molecule" and "proven niche therapy" is the whole lesson — plus a regulatory twist: the FDA has moved to remove VIP from the list of compoundable drugs.

In brief

VIP is a 28-amino-acid endogenous neuropeptide with broad, well-established physiology — it's a potent vasodilator and bronchodilator, a strong anti-inflammatory/immune regulator, and, strikingly, a master neurotransmitter of the brain's circadian clock (the SCN uses VIP to keep the body on solar time; mice without VIP lose their rhythms). Given all that, its gray-market life is surprisingly narrow: it's used mainly as a compounded nasal spray in the "CIRS / mold-illness" protocol of one physician, Ryan Shoemaker, as the final "capstone" step after upstream treatments — on the theory that biotoxin illness depletes regulatory neuropeptides. The catch: almost all the human evidence (an open-label trial of 20 patients, a 15-patient RNA-Seq study, a brain-volume study) comes from Shoemaker's own group, is small and open-label, isn't independently replicated, and addresses a diagnosis (CIRS) that mainstream medicine doesn't broadly recognise. Meanwhile the FDA has moved to pull VIP from the compounding list, and the serious drug-development action is elsewhere (the analog aviptadil in ARDS/COVID). Honest read: a genuinely important hormone whose headline gray-market use is thinly evidenced and single-sourced — big biology, small and shaky proof for the thing it's sold for.

Legal standing, by region
European Union
not an approved consumer product

not an approved consumer product; investigational. Not a cosmetic.

United States
Compounded (Rx) where lawful

not an approved drug for CIRS or general use; historically available as a compounded nasal spray (503A) — but the FDA has moved to remove VIP from the compoundable list, clouding that route. The analog aviptadil has been investigational (ARDS/COVID), not generally approved.

Evidence, by outcome
How we grade →

An honest grade per outcome — drawn from the evidence, not any catalogue. Hype and undemonstrated marketing claims grade low.

OutcomeEvidence base · effectGrade
Endogenous physiology (circadian/SCN, vasodilation, anti-inflammatory)
This grades the molecule's natural role, NOT any benefit of taking exogenous VIP. "VIP is important in the body" ≠ "VIP spray treats your condition"
Extensive, well-replicated basic science (VIP is a real, central hormone)
A
CIRS / mold-illness ("capstone" nasal-spray therapy — the marketed use)
Almost entirely single-investigator (Shoemaker), open-label, small, unreplicated; CIRS is a contested diagnosis. Reported safety over long use is the strongest point
Open-label 20-pt trial (18+ mo), 15-pt RNA-Seq, grey-matter-volume study
D
Inflammatory / pulmonary disease (inhaled VIP; aviptadil in ARDS/COVID)
Real drug-development interest — but not established/approved; results mixed/inconclusive
Legitimate research interest; aviptadil trials
C
Circadian / sleep, anxiety/depression, "anti-aging," nootropic (speculative gray-market)
No controlled human trials for these self-use claims; extrapolating from VIP's natural roles is unjustified
Association studies + strong basic biology, but no interventional human proof
F
Safety
Reported well-tolerated in the CIRS setting; but it's a potent vasoactive/immune hormone, off-protocol self-dosing is unstudied, and product quality is unverified
Long CIRS-protocol use reported
Disclosure

Vallydia sells its own cosmetic serums, and some ingredients graded here belong to the same categories as those products. Grades are drawn from the published evidence by the method we publish, and applied to our own ingredients on the same terms — our copper-peptide serum is graded no more kindly than the peptides it competes with. We disclose the interest so you can weigh it.

Trade names shown here (for example Matrixyl, Argireline, Syn-Ake) are the property of their respective owners and are used only to identify the ingredient under discussion. Their appearance implies no affiliation with, or endorsement by, the proprietor.

Evidence changes

Get notified if this changes

We track new research and update these grades as the evidence moves. Leave your email and we'll tell you if the evidence for VIP (Vasoactive Intestinal Peptide) changes - nothing else.

One ingredient, one purpose. No marketing, no sharing. Unsubscribe anytime. See our privacy policy.

Identity

a 28-amino-acid endogenous neuropeptide of the secretin/glucagon family, first isolated (Said & Mutt, ~1970) from intestine — hence the name — but in fact distributed body-wide: brain, gut, lungs, pancreas, immune system, vasculature. It signals through VPAC1/VPAC2 receptors (GPCRs, cAMP). Unlike most register entries (synthetic or gray-market-only), VIP is a genuine human hormone with broad, textbook physiology — which is exactly what makes its narrow gray-market positioning notable.

Mechanism (as proposed)

VIP signals through VPAC1 and VPAC2 receptors (G-protein-coupled, raising cAMP). Its natural actions are wide: relaxing vascular and airway smooth muscle (vasodilation/bronchodilation), down-regulating innate immune/inflammatory responses (shifting cytokine balance, calming over-active innate immunity), providing neuroprotection, and — in the suprachiasmatic nucleussynchronising the cellular circadian oscillators (the CLOCK/BMAL1–PER/CRY feedback loop) to environmental light via ERK1/2 signalling. In the CIRS framework, the proposed therapeutic logic is replacement: if regulatory neuropeptides are depleted by biotoxin illness, restoring VIP provides the "capstone" regulatory signal that lets the inflammatory cascade resolve — but note this framework's clinical validation is exactly what's limited. The biology is robust; the niche-therapeutic claim is not (yet) independently substantiated.

Sources — 5 cited
01Hamnett R, et al. Vasoactive intestinal peptide controls the suprachiasmatic circadian clock network via ERK1/2 and DUSP4. Nat Commun. 2019 (circadian master-clock role).
02Smalley SG, Barrow PA, Foster N. Immunomodulation of innate immune responses by VIP: therapeutic potential in inflammatory disease. Clin Exp Immunol. 2009 (PMID 19604262).
03Shoemaker RC, et al. VIP corrects chronic inflammatory response syndrome (CIRS) acquired following exposure to water-damaged buildings. Health. 2013 (open-label, 20 patients) — the primary CIRS reference; plus RNA-Seq (Med Res Arch 2016) and grey-matter-volume (Internal Medicine Review 2017). ⚠ Predominantly single-investigator, open-label, unreplicated.
04Vu JP, et al. Regulation of appetite, body composition, and metabolic hormones by VIP. J Mol Neurosci. 2015.
05FDA compounding-list action re: VIP (removal announced); aviptadil (RLF-100) ARDS/COVID trials (context). CIRS is a contested diagnosis in mainstream medicine.
Updated 2026-07-13 (watch: FDA compounding status, and whether any independent (non-Shoemaker) controlled trial of intranasal VIP in CIRS or inflammatory disease appears — that would be decisive)

Grades reflect the published evidence, not our interest. No dosing, reconstitution, or administration is published for research compounds — that restraint is deliberate.

Related compounds
CerebrolysinC
Peptide
ThymalinC
Peptide
Afamelanotide (Scenesse / Melanotan-1)A
Peptide
Melanotan IIC
Peptide
PT-141 (Bremelanotide)B
Peptide
Explore by goal
Neuro & cognitiveAnti-inflammatorySleep & circadian
Vallydia

A neutral reference and a lawful-lane shop. Information for those who seek it — never promotion.

RegionInternational
ExploreRegisterThe Register — full indexCategoriesTrust & COAHow we gradeOpen dataBrands
ShopCosmetic peptidesJournalQuizzes
TermsPrivacyCookiesReturnsShippingImprint

This site provides neutral scientific reference and sells only products lawful in your region. Nothing here is medical advice, a recommendation, or an offer to supply unapproved medicines. No dosing or administration is published for research compounds. Cosmetic peptides per Regulation (EC) 1223/2009. Unapproved injectable peptides are neither sold nor advertised in the EU (Directive 2001/83/EC, Title VIII). © 2026 Vallydia.